Comparison

Cagrilintide vs tirzepatide

Cagrilintide and tirzepatide are both once-weekly injections studied for weight, but they work through different hormone systems and sit at different regulatory stages. Cagrilintide is an amylin analog, tirzepatide is a GLP-1/GIP incretin, and only tirzepatide is FDA-approved, so the evidence behind each is not on equal footing.

Reviewed for accuracy · Last reviewed July 8, 2026

Side by side

CagrilintideTirzepatide
Hormone systemAmylin (long-acting amylin receptor agonist)Incretin (GLP-1 and GIP)
Route and frequencySubcutaneous, once weeklySubcutaneous, once weekly
Doses studied or labeled0.3 – 4.5 mg weekly (Phase 2 monotherapy)2.5 – 15 mg (labeled titration)
Approval statusInvestigational, not FDA-approvedFDA-approved (Mounjaro, Zepbound)
Evidence basePhase 2 obesity trial; Phase 3 for the semaglutide combination (CagriSema)Phase 3 trial data and a product label

Which is right for you

The clearest practical difference is regulatory. Tirzepatide has an approved label, a defined titration, and Phase 3 evidence, whereas cagrilintide is investigational: its monotherapy human evidence comes from a Phase 2 dose-finding trial, with Phase 3 data centered on the semaglutide combination (CagriSema) rather than cagrilintide alone.

Mechanistically these are different kinds of drug. Cagrilintide mimics amylin, a hormone that signals fullness and slows gastric emptying, while tirzepatide acts on the GLP-1 and GIP incretin receptors. Because they target separate pathways, cagrilintide has been studied paired with a GLP-1 drug rather than as a direct incretin substitute. Whether either approach is preferable in practice is not something the current evidence lets anyone state as fact.

Both were studied as once-weekly subcutaneous injections with gradual dose escalation, and both reported predominantly dose-related gastrointestinal side effects such as nausea. Neither of these summaries is a substitute for medical advice about which, if either, is appropriate.

FAQ

Is cagrilintide the same kind of drug as tirzepatide?No. Cagrilintide is an amylin analog, targeting the amylin pathway, while tirzepatide is an incretin acting on GLP-1 and GIP. Because they work through different hormone systems, cagrilintide has been studied combined with a GLP-1 drug (CagriSema).
Is cagrilintide approved like tirzepatide?No. Tirzepatide is FDA-approved (as Mounjaro and Zepbound). Cagrilintide is investigational with no FDA-approved product; its Phase 3 evidence centers on the semaglutide combination CagriSema, which was under review as of 2026.

References

  1. Once-Weekly Cagrilintide for Weight Management in People With Overweight and Obesity: A Dose-Finding Phase 2 TrialThe Lancet · 2021 · PMID 34798060 · DOI 10.1016/S0140-6736(21)01751-7 · NCT03856047
  2. Cagrilintide-Semaglutide in Adults With Overweight or Obesity and Type 2 Diabetes (REDEFINE 2)New England Journal of Medicine · 2025 · PMID 40544432 · DOI 10.1056/NEJMoa2502082 · NCT05394519
  3. Investigation of Safety and Efficacy of NNC0174-0833 for Weight Management: A Dose-Finding TrialClinicalTrials.gov (sponsor: Novo Nordisk A/S) · 2019 · NCT03856047
  4. Tirzepatide Once Weekly for the Treatment of Obesity (SURMOUNT-1)New England Journal of Medicine · 2022 · PMID 35658024 · DOI 10.1056/NEJMoa2206038
  5. MOUNJARO (tirzepatide) injection: DailyMed labelDailyMed (U.S. National Library of Medicine) · current · DailyMed setid d2d7da5d-ad07-4228-955f-cf7e355c8cc0
  6. ZEPBOUND (tirzepatide) injection: DailyMed labelDailyMed (U.S. National Library of Medicine) · current · DailyMed setid 487cd7e7-434c-4925-99fa-aa80b1cc776b

This page is an independent educational reference and is not medical advice, and does not indicate any approval status for any use. Talk to a doctor before starting any compound.